SCHEMBL7778714

SCHEMBL7778714

CC(N)c1ccc(C#N)cc1.CC(N)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.59
PDE2A O00408 2/20 0.51
CYP19A1 P11511 5/20 0.45
CYP3A4 P08684 1/20 0.42
CYP3A5 P20815 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.40
ADRB2 P07550 1/20 0.38
PTPN5 P54829 1/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
ALOX15 P16050 1/20 0.37
BRCA1 P38398 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
DGAT1 O75907 1/20 0.37
SOAT1 P35610 1/20 0.37
KCNH2 Q12809 1/20 0.37
CYP2A6 P11509 1/20 0.36
DHODH Q02127 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7575723 0.87 TAAR1 (0.55) KIF11PDE2ACYP19A1CYP2A6VNN1
SCHEMBL7575719 0.86 KIF11 (0.45) KIF11PDE2ACYP19A1CYP3A4CYP3A5
SCHEMBL12230784 0.86 KIF11 (0.63) KIF11PDE2ACYP19A1CYP3A4CYP3A5
SCHEMBL12230783 0.86 KIF11 (0.63) KIF11PDE2ACYP19A1CYP3A4CYP3A5
SCHEMBL12230279 0.86 KIF11 (0.63) KIF11PDE2ACYP19A1CYP3A4CYP3A5
SCHEMBL268077 0.85 PDE2A (0.67) KIF11PDE2AADRB2ALDH1A1
SCHEMBL701658 0.85 PDE2A (0.67) KIF11PDE2AADRB2ALDH1A1
SCHEMBL335039 0.85 PDE2A (0.67) KIF11PDE2AADRB2ALDH1A1
SCHEMBL320272 0.85 ADRB2 (0.50) PDE2ACYP19A1CYP3A4ADRB2ALDH1A1
SCHEMBL319930 0.85 ADRB2 (0.50) PDE2ACYP19A1CYP3A4ADRB2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144397-A3 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP Wyeth (US) 2002-09-11 EP disclosed
EP-1144397-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-17 EP disclosed
WO-2000034258-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed