SCHEMBL7778751

SCHEMBL7778751

OC(CNCCOc1cc2[nH]c3ccccc3c2cc1[AsH2])c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.49
ADRB1 P08588 6/20 0.46
DRD2 P14416 5/20 0.46
ADRB3 P13945 5/20 0.46
DRD1 P21728 3/20 0.46
DRD4 P21917 3/20 0.46
DRD3 P35462 3/20 0.46
TLR4 O00206 2/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 2/20 0.46
SLC22A2 O15244 1/20 0.46
SLC22A1 O15245 1/20 0.46
MLNR O43193 1/20 0.46
NR1I2 O75469 1/20 0.46
KCNK2 O95069 1/20 0.46
ABCB11 O95342 1/20 0.46
APP P05067 1/20 0.46
ABCB1 P08183 1/20 0.46
HTR1A P08908 1/20 0.46
ADRA2A P08913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7068691 0.88 ADRB2 (0.50) ADRB2ADRB1DRD2ADRB3DRD1
SCHEMBL7070286 0.87 ADRB2 (0.49) ADRB2ADRB1DRD2ADRB3DRD1
Hydrochloric Acid SCHEMBL7107109 0.86 ADRB2 (0.48) ADRB2ADRB1DRD2ADRB3DRD1
SCHEMBL6905931 0.82 ALOX15 (0.54) ADRB2ADRB1ADRB3KDM4EADRA1A
SCHEMBL6912018 0.82 ALOX15 (0.54) ADRB2ADRB1ADRB3KDM4EADRA1A
SCHEMBL6912318 0.82 ALOX15 (0.54) ADRB2ADRB1ADRB3KDM4EADRA1A
SCHEMBL7069436 0.82 ADRB2 (0.47) ADRB2ADRB1DRD2ADRB3DRD1
Hydrochloric Acid SCHEMBL7113305 0.81 ALOX15 (0.56) ADRB2ADRB1ADRB3ADRA1AALDH1A1
Hydrochloric Acid SCHEMBL7111563 0.81 ALOX15 (0.56) ADRB2ADRB1ADRB3ADRA1AALDH1A1
Hydrochloric Acid SCHEMBL7108157 0.81 ALOX15 (0.56) ADRB2ADRB1ADRB3ADRA1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1128845-A1 COMBINATIONS COMPRISING A BETA-AGONIST AND A FURTHER ANTDIABETIC AGENT SMITHKLINE BEECHAM PLC (GB) 2001-09-05 EP disclosed
WO-2000027434-A1 COMBINATIONS COMPRISING A BETA-AGONIST AND A FURTHER ANTIDIABETIC AGENT SMITHKLINE BEECHAM P.L.C. (GB) 2000-05-18 WO disclosed