SCHEMBL7779256

SCHEMBL7779256

COC(=O)COc1nc(N)c(Cl)cc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.43
KDM4E B2RXH2 2/20 0.40
GLA P06280 1/20 0.40
CFTR P13569 4/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
PTK2 Q05397 1/20 0.37
PDK2 Q15119 1/20 0.37
AR P10275 1/20 0.37
HTT P42858 1/20 0.36
PDGFRB P09619 1/20 0.36
KDR P35968 1/20 0.36
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
NOTUM Q6P988 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11611002 0.84 LMNA (0.54) LMNAKDM4EKMT2AMAPTHTT
SCHEMBL7779272 0.79 CFTR (0.44) KDM4EGLACFTRMAPTCYP1A2
SCHEMBL7779192 0.77 CFTR (0.40) CFTRMAPTKDRCYP1A2CYP2C19
SCHEMBL7779269 0.73 CDK1 (0.39) LMNACFTRKDR
SCHEMBL31711403 0.71 CDK1 (0.36) CFTRMAPTCYP1A2CYP2C19
SCHEMBL11611738 0.70 TSHR (0.40) LMNAKDM4EKMT2A
SCHEMBL11563321 0.70 LMNA (0.54) LMNAKDM4EKMT2AMAPTPDK2
SCHEMBL3232675 0.69 LMNA (0.57) LMNAKDM4EKMT2AMAPTHTT
SCHEMBL31438450 0.69 LMNA (0.57) LMNAKDM4EKMT2AMAPTHTT
SCHEMBL8531219 0.68 AURKA (0.39) LMNACFTRMAPTKDRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759429-B1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF AG (DE) 2001-10-24 EP claimed
US-5750705-A HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1998-05-12 US claimed
EP-0759429-A1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF Aktiengesellschaft (DE) 1997-02-26 EP claimed