SCHEMBL7779192

SCHEMBL7779192

COc1nc(N)c(Cl)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.40
AURKA O14965 2/20 0.37
KDR P35968 2/20 0.37
AURKB Q96GD4 2/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
DYRK1A Q13627 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPT P10636 1/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
RORB Q92753 1/20 0.33
IDO1 P14902 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8531219 0.86 AURKA (0.39) CFTRAURKAKDRAURKBGSK3A
SCHEMBL7779272 0.82 CFTR (0.44) CFTRCYP1A2CYP3A4CYP2C19MAPT
SCHEMBL31711403 0.82 CDK1 (0.36) CFTRCYP1A2CYP3A4CYP2C19MAPT
SCHEMBL7779256 0.77 LMNA (0.43) CFTRKDRCYP1A2CYP2C19MAPT
SCHEMBL31717937 0.76 PIK3CD (0.41) IDO1
SCHEMBL7784302 0.76 PIK3CD (0.41) IDO1
SCHEMBL7779269 0.75 CDK1 (0.39) CFTRKDRIDO1
SCHEMBL6953346 0.75 KMT2A (0.38) AURKAKDRAURKBCYP1A2CYP3A4
SCHEMBL8007192 0.74 GSK3A (0.40) GSK3AGSK3BDYRK1ACLK4CYP3A4
SCHEMBL7786072 0.74 MPL (0.35) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759429-B1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF AG (DE) 2001-10-24 EP claimed
US-5750705-A HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1998-05-12 US claimed
EP-0759429-A1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF Aktiengesellschaft (DE) 1997-02-26 EP claimed
EP-0759429-B1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF AG (DE) 2001-10-24 EP disclosed
US-6252069-B1 REACTING ANTHRANILIC ISOPROPAMIDE WITH SULFUR TRIOXIDE BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
US-5849920-A Substituted trifluoromethylpyridines BASF AKTIENGESELLSCHAFT (DE) 1998-12-15 US disclosed
US-5750705-A HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1998-05-12 US disclosed
EP-0759429-A1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF Aktiengesellschaft (DE) 1997-02-26 EP disclosed