SCHEMBL7784332

SCHEMBL7784332

COc1ccc2c(c1)C(CCNC(C)=O)=CC2

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 15/20 0.78
MTNR1B P49286 15/20 0.78
NQO2 P16083 5/20 0.78
SMN1; SMN2 Q16637 1/20 0.52
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1289437 0.89 MTNR1A (0.62) MTNR1AMTNR1BNQO2SMN1; SMN2HTR2C
SCHEMBL30589884 0.89 MTNR1A (0.62) MTNR1AMTNR1BNQO2SMN1; SMN2HTR2C
SCHEMBL7784380 0.88 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7785010 0.85 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7779922 0.85 MTNR1A (0.83) MTNR1AMTNR1BNQO2
SCHEMBL7787100 0.81 MTNR1A (0.54) MTNR1AMTNR1BNQO2
SCHEMBL7786940 0.81 MTNR1A (0.53) MTNR1AMTNR1BNQO2
SCHEMBL8349133 0.79 NQO2 (0.62) MTNR1AMTNR1BNQO2HTR2C
SCHEMBL7784524 0.79 MTNR1A (0.50) MTNR1AMTNR1BNQO2
SCHEMBL7820683 0.78 NQO2 (0.61) MTNR1AMTNR1BNQO2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848699-B1 BENZOCYCLOALKENE COMPOUNDS WITH MELATONINE RECEPTOR BINDING AFFINITY, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-24 EP disclosed
US-5922771-A MELATONIN RECEPTOR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-13 US disclosed
EP-0848699-A1 BENZOCYCLOALKENE COMPOUNDS WITH MELATONINE RECEPTOR BINDING AFFINITY, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-06-24 EP disclosed
WO-1997005098-A1 BENZOCYCLOALKENE COMPOUNDS WITH MELATONINE RECEPTOR BINDING AFFINITY, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-02-13 WO disclosed