SCHEMBL7784544

SCHEMBL7784544

Clc1ccc([N]C2CCCCCC2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 2/20 0.41
HTR3B O95264 2/20 0.41
HTR3A P46098 2/20 0.41
HTR3D Q70Z44 2/20 0.41
HTR3C Q8WXA8 2/20 0.41
MAPK1 P28482 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
SLC6A3 Q01959 7/20 0.39
KMT2A Q03164 2/20 0.38
SLC6A4 P31645 4/20 0.38
SLC6A2 P23975 2/20 0.38
KCNH2 Q12809 2/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 3/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
ALOX12 P18054 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790021 0.81 HTR3E (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL28279936 0.74 MAPK1 (0.65) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7794524 0.74 KDM4E (0.37) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7793294 0.73 HTR3E (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7794041 0.69 NPC1 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9861135 0.69 KMT2A (0.57) MAPK1SLC6A3KMT2AMAPTALOX12
SCHEMBL9861146 0.69 KMT2A (0.57) MAPK1SLC6A3KMT2AMAPTALOX12
SCHEMBL723225 0.69 ALDH1A1 (0.39) KMT2AMAPT
SCHEMBL7418307 0.67 SLC22A2 (0.37) TDP1KMT2AMAPTMEN1LMNA
SCHEMBL2478208 0.67 CYP1A2 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed