SCHEMBL7785072

SCHEMBL7785072

COc1ccc(C(NC(C)c2ccc(F)c(F)c2)c2ccc(F)c(N)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
HTT P42858 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
ACHE P22303 1/20 0.37
APP P05067 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 2/20 0.36
CASR P41180 2/20 0.36
KMT2A Q03164 4/20 0.36
MITF O75030 1/20 0.36
ACP3 P15309 2/20 0.34
TP53 P04637 1/20 0.34
ADRB2 P07550 1/20 0.33
ALOX5 P09917 1/20 0.33
NFE2L2 Q16236 1/20 0.33
PDPK1 O15530 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27540176 0.90 ALDH1A1 (0.39) ALDH1A1MAPTHTTL3MBTL1CA1
SCHEMBL7785536 0.90 ALDH1A1 (0.39) ALDH1A1MAPTHTTL3MBTL1CA1
SCHEMBL7780785 0.90 TDP1 (0.43) ALDH1A1MAPTHTTL3MBTL1CA1
SCHEMBL7780640 0.86 ALDH1A1 (0.41) ALDH1A1MAPTHTTL3MBTL1CA1
SCHEMBL7785127 0.86 ALDH1A1 (0.41) ALDH1A1MAPTHTTL3MBTL1CA1
SCHEMBL7780432 0.86 ALDH1A1 (0.41) ALDH1A1MAPTHTTL3MBTL1CA1
SCHEMBL7784893 0.86 ALDH1A1 (0.34) ALDH1A1MAPTHTTL3MBTL1CA1
SCHEMBL7780568 0.84 ALDH1A1 (0.39) ALDH1A1MAPTHTTL3MBTL1CA1
SCHEMBL7784903 0.82 ALDH1A1 (0.37) ALDH1A1MAPTHTTL3MBTL1CA1
Hydrochloric Acid SCHEMBL7780344 0.82 ALDH1A1 (0.44) ALDH1A1MAPTHTTL3MBTL1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed