SCHEMBL7784903

SCHEMBL7784903

COc1ccc(C(NC(C)c2ccc(F)c(F)c2)c2cc(N)ccc2F)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
MAPT P10636 2/20 0.37
HTT P42858 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
MAPK1 P28482 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
ACHE P22303 1/20 0.35
APP P05067 2/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 2/20 0.35
GAA P10253 2/20 0.35
CYP3A4 P08684 1/20 0.35
NR4A1 P22736 1/20 0.34
KMT2A Q03164 4/20 0.33
ACP3 P15309 2/20 0.33
TP53 P04637 1/20 0.33
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7787455 0.92 CYP2D6 (0.39) ALDH1A1MAPTHTTL3MBTL1TDP1
SCHEMBL7780785 0.90 TDP1 (0.43) ALDH1A1MAPTHTTL3MBTL1TDP1
SCHEMBL7780432 0.84 ALDH1A1 (0.41) ALDH1A1MAPTHTTL3MBTL1TDP1
SCHEMBL7780640 0.84 ALDH1A1 (0.41) ALDH1A1MAPTHTTL3MBTL1TDP1
SCHEMBL7780568 0.84 ALDH1A1 (0.39) ALDH1A1MAPTHTTL3MBTL1TDP1
SCHEMBL7785127 0.84 ALDH1A1 (0.41) ALDH1A1MAPTHTTL3MBTL1TDP1
SCHEMBL7780363 0.83 CA1 (0.34) ALDH1A1MAPTCA1CA2ACHE
SCHEMBL7785072 0.82 ALDH1A1 (0.38) ALDH1A1MAPTHTTL3MBTL1TDP1
SCHEMBL7787479 0.81 MEN1 (0.39) ALDH1A1MAPK1CA1CA2ACHE
SCHEMBL7785020 0.81 GAA (0.40) ALDH1A1MAPTHTTL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed