SCHEMBL7785708

SCHEMBL7785708

O=C(O)CC(NS(=O)(=O)c1ccccc1)c1cccc(NS(=O)(=O)c2cccc(NC3=NCCN3)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.53
ITGAV P06756 14/20 0.53
ITGA2B P08514 3/20 0.52
ITGB1 P05556 2/20 0.47
ITGB5 P18084 2/20 0.47
EEF2K O00418 3/20 0.44
ALDH1A1 P00352 1/20 0.42
ATM Q13315 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ITGA5 P08648 1/20 0.41
ITGB6 P18564 1/20 0.41
ITGB8 P26012 1/20 0.41
ITGA8 P53708 1/20 0.41
OGT O15294 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8357385 0.86 ITGB3 (0.55) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL6798729 0.83 ITGB3 (0.44) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7997106 0.81 ITGB3 (0.70) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7856513 0.79 ITGB3 (0.45) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL3835113 0.78 HTR6 (0.57) ITGB3ITGAVEEF2KALDH1A1ATM
SCHEMBL2841846 0.73 ITGB3 (0.59) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL6367424 0.73 ITGB3 (0.61) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL6366667 0.73 ITGB3 (0.60) ITGB3ITGAVEEF2KALDH1A1ATM
SCHEMBL7786198 0.71 ITGB3 (0.49) ITGB3ITGAVEEF2KALDH1A1ATM
SCHEMBL2837308 0.71 ITGB3 (0.53) ITGB3ITGAVITGA2BITGB1ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147079-A2 BETA-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS Bayer Aktiengesellschaft (DE) 2001-10-24 EP disclosed
US-6291503-B1 β-phenylalanine derivatives as integrin antagonists BAYER AKTIENGESELLSCHAFT (DE) 2001-09-18 US disclosed
WO-2000041469-A2 β-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2000-07-20 WO disclosed