SCHEMBL7786876

SCHEMBL7786876

CCCCCC(CCCC)CC(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 9/20 0.61
FFAR1 O14842 2/20 0.48
FFAR4 Q5NUL3 1/20 0.48
LMNA P02545 1/20 0.48
PPARD Q03181 3/20 0.47
MAPT P10636 1/20 0.47
LCK P06239 1/20 0.47
ZDHHC20 Q5W0Z9 1/20 0.47
ZDHHC2 Q9UIJ5 1/20 0.47
AKR1B1 P15121 1/20 0.46
CA2 P00918 2/20 0.45
MAPK1 P28482 1/20 0.45
PPARG P37231 2/20 0.44
PPARA Q07869 2/20 0.44
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44
SLC22A6 Q4U2R8 1/20 0.44
SLC22A8 Q8TCC7 1/20 0.44
TLR2 O60603 1/20 0.44
HDAC11 Q96DB2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18187980 0.98 GPR84 (0.64) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL9500560 0.98 GPR84 (0.64) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL6837132 0.98 GPR84 (0.64) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL18188038 0.98 GPR84 (0.64) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL18187989 0.98 GPR84 (0.64) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL18187992 0.98 GPR84 (0.64) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL10438737 0.98 GPR84 (0.64) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL4597758 0.98 GPR84 (0.63) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL5362865 0.98 GPR84 (0.57) GPR84FFAR1FFAR4LMNAPPARD
SCHEMBL23879500 0.95 GPR84 (0.67) GPR84FFAR1FFAR4LMNAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3632994-B1 OIL-BASED INKJET INK RISO KAGAKU CORP (JP) 2024-01-24 EP claimed
US-20260109911-A1 FRICTION MODIFIER FOR WET CLUTCH CHEVRON ORONITE CO (US) 2026-04-23 US disclosed
WO-2024220394-A1 FRICTION MODIFIER FOR AUTOMATIC TRANSMISSION FLUID CHEVRON ORONITE COMPANY LLC (US) 2024-10-24 WO disclosed
WO-2024220396-A1 FRICTION MODIFIER FOR WET CLUTCH CHEVRON ORONITE COMPANY LLC (US) 2024-10-24 WO disclosed
CN-103443099-B Regulate composition and the method for FXR NOVARTIS AG (CH) 2016-03-23 CN disclosed
CN-103443099-A Compositions and methods for modulating FXR IRM LLC 2013-12-11 CN disclosed
CN-1407982-A Serotonergic benzofurans LILLY CO ELI (US) 2003-04-02 CN disclosed
US-6251903-B1 Alkyl, azido, alkoxy, and fluoro-substituted and fused quinoxalinediones and the use thereof as glycine receptor antagonist COCENSYS, INC. 2001-06-26 US disclosed
US-6147075-A ANALGESICS; PSYCHOLOGICAL DISORDERS COCENSYS, INC. (US) 2000-11-14 US disclosed
US-5977107-A Alkyl, azido, alkoxy, and fluoro-substituted and fused quinoxalinediones and the use thereof as glycine receptor antagonists COCENSYS, INC. (US) 1999-11-02 US disclosed
US-5863916-A 8-aza, 6-aza and 6,8-diaza-1,4-dihydroquinoxaline-2,3-diones and the use thereof as antagonists for the glycine/NMDA receptor STATE OF OREGON, ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER-EDUCATION, ACTING FOR AND ON BEHALF OF THE OREGON HEALTH SCIENCES UNIVERSITY AND THE UNIVERSITY OF OREGON (US) 1999-01-26 US disclosed
US-5856476-A Processes for preparing azepiones useful as intermediates in the preparation of inhibitors of angiotensin converting enzyme and neutral endopeptidase E. R. SQUIBBS & SONS, INC. (US) 1999-01-05 US disclosed
US-5723457-A COMPOUMDS FOR CARDIOVASCULAR DISORDERS AND INHIBITORS OF ANGIOTENSIN CONVERTING ENZYMES E. R. SQUIBB & SONS, INC. (US) 1998-03-03 US disclosed
US-5631373-A NERVOUS SYSTEM DISORDERS STATE OF OREGON, ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION, ACTING FOR AND ON BEHALF OF THE OREGON HEALTH SCIENCES UNIVERSITY AND THE UNIVERSITY OF OREGON, EUGENE OREGON (US) 1997-05-20 US disclosed
US-5622952-A NERVOUS SYSTEM DISORDERS; ADMINISTERING 1,4-DIHYDROQUINOXALINE-2,3-DIONE STATE OF OREGON, ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION, ACTING FOR AND ON BEHALF OF THE OREGON HEALTH SCIENCES UNIVERSITY AND THE UNIVERSITY OF OREGON, EUGENE OREGON (US) 1997-04-22 US disclosed
US-5620978-A 8-aza, 6-aza and 6,8-diaza-1,4-dihydroquinoxaline-2,3-diones and the use thereof as antagonists for the glycine/NMDA receptor STATE OF OREGON, ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION, ACTING FOR AND ON BEHALF OF THE OREGON HEALTH SCIENCES UNIVERSITY AND THE UNIVERSITY OF OREGON, EUGENE OREGON (US) 1997-04-15 US disclosed
US-5620979-A TREATING NEURONAL LOSS ASSOCIATED WITH STROKE, ISCHEMIA, CENTRAL NERVOUS SYSTEM TRAUMA, HYPOGLYCEMIA OR SURGERY STATE OF OREGON, ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION, ACTING FOR AND ON BEHALF OF THE OREGON HEALTH SCIENCES UNIVERSITY AND THE UNIVERSITY OF OREGON, EUGENE OREGON (US) 1997-04-15 US disclosed
US-5514680-A ANTICONVULSANTS WITH 5,6,7-TRISUBSTITUTED-1,4-DIHYDROQUINOXALINE-2,3-DIONE THE STATE OF OREGON, ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION, ACTING FOR AND ON BEHALF OF THE OREGON HEALTH SCIENCES UNIVERSITY (US) 1996-05-07 US disclosed
WO-1994000124-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF WEBER ECKARD (US) 1994-01-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260109911-A1 FRICTION MODIFIER FOR WET CLUTCH SMCHD1, CLTC, CLTA GPR84 2785/4885FFAR1 1792/4885FFAR4 1362/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.