SCHEMBL7786992

SCHEMBL7786992

O=C(NC(CO)Cc1ccccc1)c1cccc(C=Cc2ccc3ccccc3c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 11/20 0.53
CAPN1 P07384 2/20 0.52
CTSL P07711 1/20 0.49
CTSB P07858 1/20 0.49
ROCK2 O75116 1/20 0.48
RPS6KA5 O75582 1/20 0.48
RPS6KA4 O75676 1/20 0.48
PRKACA P17612 1/20 0.48
MAPK1 P28482 1/20 0.48
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48
IRAK1 P51617 1/20 0.48
PRKX P51817 1/20 0.48
ROCK1 Q13464 1/20 0.48
PRKG1 Q13976 1/20 0.48
PKN2 Q16513 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
SGK2 Q9HBY8 1/20 0.48
CTRB1 P17538 1/20 0.47
F10 P00742 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7787838 0.91 MAPK1 (0.56) PIN1CAPN1CTSLCTSBROCK2
SCHEMBL7787781 0.84 CAPN1 (0.72) PIN1CAPN1CTSLCTSBF10
SCHEMBL7789913 0.83 CAPN1 (0.74) PIN1CAPN1CTSLCTSBROCK2
SCHEMBL7789911 0.83 CAPN1 (0.74) PIN1CAPN1CTSLCTSBROCK2
SCHEMBL7782138 0.80 NPC1 (0.59) PIN1ROCK2RPS6KA5RPS6KA4PRKACA
SCHEMBL14005615 0.80 HPGDS (0.58) PIN1CTSLROCK2RPS6KA5RPS6KA4
SCHEMBL6800557 0.79 CAPN1 (0.54) PIN1CAPN1CTSLCTSBROCK2
SCHEMBL3682310 0.78 CTRB1 (0.73) PIN1CTSLROCK2RPS6KA5RPS6KA4
SCHEMBL5685800 0.78 CTRB1 (0.73) PIN1CTSLROCK2RPS6KA5RPS6KA4
SCHEMBL3682311 0.78 CTRB1 (0.73) PIN1CTSLROCK2RPS6KA5RPS6KA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed