SCHEMBL7787640

SCHEMBL7787640

O=C(c1ccncc1)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.68
CES2 O00748 1/20 0.62
CES1 P23141 1/20 0.62
TP53 P04637 1/20 0.60
ALDH1A1 P00352 2/20 0.58
TSHR P16473 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.57
POLB P06746 1/20 0.57
CACNA1B Q00975 1/20 0.57
APBA1 Q02410 1/20 0.57
LMNA P02545 3/20 0.56
KMT2A Q03164 5/20 0.56
MEN1 O00255 3/20 0.56
HPGD P15428 1/20 0.55
ATM Q13315 1/20 0.55
MAPT P10636 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
RXFP1 Q9HBX9 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridine SCHEMBL28090680 0.91 TP53 (0.61) L3MBTL1CES2CES1TP53ALDH1A1
SCHEMBL181572 0.88 CES2 (0.78) CES2CES1TP53ALDH1A1TSHR
Pyrimidine SCHEMBL27895077 0.88 TP53 (0.61) L3MBTL1CES2CES1TP53ALDH1A1
SCHEMBL333455 0.86 TP53 (0.73) L3MBTL1CES2CES1TP53ALDH1A1
SCHEMBL8962468 0.86 CES2 (0.75) CES2CES1TP53ALDH1A1TSHR
SCHEMBL11295596 0.85 TP53 (0.71) L3MBTL1CES2CES1TP53ALDH1A1
SCHEMBL3234327 0.85 CES2 (0.68) L3MBTL1CES2CES1TP53ALDH1A1
Ammonia Solution, Strong SCHEMBL27493385 0.85 TP53 (0.71) L3MBTL1CES2CES1TP53ALDH1A1
Iodide SCHEMBL28290571 0.85 TP53 (0.71) L3MBTL1CES2CES1TP53ALDH1A1
Bromide SCHEMBL28137305 0.85 TP53 (0.71) L3MBTL1CES2CES1TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed
EP-0046446-A1 Polyazaheterocyclic compounds, process for their preparation and pharmaceutical compositions containing them CIBA-GEIGY AG (CH) 1982-02-24 EP disclosed