SCHEMBL7787801

SCHEMBL7787801

O=C[C@H](Cc1ccccc1)NC(=O)c1ccc(CSc2ccc3ccccc3c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 11/20 0.58
CTSB P07858 2/20 0.46
PIN1 Q13526 3/20 0.44
CA2 P00918 1/20 0.43
PPARG P37231 2/20 0.42
PPARA Q07869 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7787804 1.00 CAPN1 (0.58) CAPN1CTSBPIN1CA2PPARG
SCHEMBL7787044 0.84 CAPN1 (0.57) CAPN1CTSBPIN1CA2CTSL
SCHEMBL7789879 0.83 CAPN1 (0.48) CAPN1KDM4E
SCHEMBL7789875 0.83 CAPN1 (0.48) CAPN1KDM4E
SCHEMBL7789993 0.81 NR1H4 (0.62) CAPN1PIN1PPARG
SCHEMBL7790056 0.81 CAPN1 (0.74) CAPN1CTSBPIN1CTSL
SCHEMBL7789863 0.80 CAPN1 (0.72) CAPN1PIN1
SCHEMBL7789862 0.80 CAPN1 (0.72) CAPN1PIN1
SCHEMBL7789989 0.80 NR1H4 (0.58) CAPN1PIN1KDM4EMEN1KMT2A
SCHEMBL7789992 0.80 NR1H4 (0.58) CAPN1PIN1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed