SCHEMBL7787044

SCHEMBL7787044

O=C[C@H](Cc1ccccc1)NC(=O)c1ccc(COSc2ccc3ccccc3c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 9/20 0.57
PIN1 Q13526 2/20 0.44
CTSB P07858 4/20 0.43
CA2 P00918 1/20 0.43
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
CTSL P07711 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789838 0.84 PIN1 (0.53) PIN1CA2NPC1MAPTCTSL
SCHEMBL7787801 0.84 CAPN1 (0.58) CAPN1PIN1CTSBCA2CTSL
SCHEMBL7787804 0.84 CAPN1 (0.58) CAPN1PIN1CTSBCA2CTSL
SCHEMBL7789862 0.82 CAPN1 (0.72) CAPN1PIN1NPC1MAPT
SCHEMBL7789863 0.82 CAPN1 (0.72) CAPN1PIN1NPC1MAPT
SCHEMBL7789993 0.79 NR1H4 (0.62) CAPN1PIN1
SCHEMBL7790056 0.78 CAPN1 (0.74) CAPN1PIN1CTSBCTSL
SCHEMBL7789992 0.78 NR1H4 (0.58) CAPN1PIN1NPC1MAPT
SCHEMBL7789989 0.78 NR1H4 (0.58) CAPN1PIN1NPC1MAPT
SCHEMBL7789857 0.77 NR1H4 (0.51) NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed