SCHEMBL7789813

SCHEMBL7789813

COC(=O)c1ccc(CSc2ccc3ccccc3c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.59
TP53 P04637 1/20 0.56
POLB P06746 2/20 0.55
THRB P10828 1/20 0.55
NPC1 O15118 5/20 0.54
RAB9A P51151 5/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
MAPT P10636 3/20 0.54
TSHR P16473 2/20 0.54
MAPK1 P28482 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
PDE7A Q13946 1/20 0.53
PDE7B Q9NP56 1/20 0.53
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 1/20 0.51
PTGDR2 Q9Y5Y4 1/20 0.49
LMNA P02545 2/20 0.49
HDAC3 O15379 1/20 0.48
NCOR1 O75376 1/20 0.48
HDAC1 Q13547 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28141839 0.89 CYP1A2 (0.53) CYP1A2TP53THRBNPC1RAB9A
SCHEMBL3916950 0.84 RAB9A (0.61) TP53NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL7350052 0.82 HTT (0.56) CYP1A2POLBNPC1RAB9ASMN1; SMN2
SCHEMBL7789800 0.81 POLB (0.53) POLBNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL5556586 0.80 TP53 (0.59) CYP1A2TP53NPC1RAB9ASMN1; SMN2
SCHEMBL4769320 0.78 KMT2A (0.66) CYP1A2TP53NPC1RAB9ASMN1; SMN2
SCHEMBL7164014 0.78 KMT2A (0.56) CYP1A2TP53POLBNPC1RAB9A
SCHEMBL1003761 0.77 KDM4E (0.62) POLBNPC1RAB9ATSHRALDH1A1
SCHEMBL4664711 0.76 EGFR (0.47) CYP1A2TP53THRBNPC1RAB9A
SCHEMBL7791330 0.76 RAB9A (0.62) POLBNPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
CN-1238761-A benzamide aldehydes and their use as cysteine protease inhibitors BASF AG (DE) 1999-12-15 CN disclosed