SCHEMBL7789864

SCHEMBL7789864

O=C(N[C@H](CO)Cc1ccccc1)c1cc(NS(=O)(=O)c2ccc3ccccc3c2)ccc1Br

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
ALDH1A1 P00352 2/20 0.52
PKM P14618 2/20 0.48
AKR1C3 P42330 1/20 0.46
LMNA P02545 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
F2 P00734 1/20 0.45
GAA P10253 1/20 0.44
PIN1 Q13526 2/20 0.43
PKLR P30613 1/20 0.43
PGR P06401 1/20 0.43
HDAC1 Q13547 2/20 0.43
NR1I2 O75469 1/20 0.43
GGPS1 O95749 1/20 0.43
ATM Q13315 1/20 0.42
GPR27 Q9NS67 1/20 0.42
ALOX12 P18054 1/20 0.42
CASP6 P55212 1/20 0.42
HDAC3 O15379 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789865 1.00 MEN1 (0.52) MEN1KMT2AALDH1A1PKMAKR1C3
SCHEMBL7787036 0.89 PKM (0.54) MEN1KMT2AALDH1A1PKMAKR1C3
SCHEMBL7787038 0.89 PKM (0.54) MEN1KMT2AALDH1A1PKMAKR1C3
SCHEMBL7790018 0.86 CAPN1 (0.53) MEN1KMT2AALDH1A1PKMAKR1C3
SCHEMBL7790014 0.86 CAPN1 (0.53) MEN1KMT2AALDH1A1PKMAKR1C3
SCHEMBL7789327 0.85 ALDH1A1 (0.57) MEN1KMT2AALDH1A1AKR1C3LMNA
SCHEMBL7789330 0.85 ALDH1A1 (0.57) MEN1KMT2AALDH1A1AKR1C3LMNA
SCHEMBL7791333 0.83 AKR1C3 (0.54) MEN1KMT2AALDH1A1AKR1C3LMNA
SCHEMBL7791335 0.83 AKR1C3 (0.54) MEN1KMT2AALDH1A1AKR1C3LMNA
SCHEMBL7786988 0.83 BCL2 (0.51) MEN1KMT2AF2PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed