SCHEMBL7790181

SCHEMBL7790181

O=C(CBr)CN(CCc1ccccc1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.51
MEN1 O00255 1/20 0.51
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
KMT2A Q03164 1/20 0.51
CA12 O43570 5/20 0.46
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
ALOX5 P09917 3/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
CA4 P22748 3/20 0.43
RCE1 Q9Y256 1/20 0.43
HDAC1 Q13547 2/20 0.42
HDAC3 O15379 1/20 0.42
MAPK1 P28482 1/20 0.42
ADRA1A P35348 1/20 0.42
HDAC4 P56524 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6359725 0.82 TDP1 (0.58) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL5933377 0.82 TDP1 (0.66) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL7796988 0.78 L3MBTL1 (0.47) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL7228409 0.78 MEN1 (0.61) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL2315734 0.77 RCE1 (0.52) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL4731326 0.75 TDP1 (0.58) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL2479873 0.75 LMNA (0.59) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL4467147 0.73 RCE1 (0.52) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL1901574 0.73 RCE1 (0.52) TDP1MEN1NPC1RAB9AKMT2A
SCHEMBL7076078 0.73 HDAC1 (0.64) TDP1NPC1RAB9AALOX5L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159260-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000055124-A2 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed