SCHEMBL7790301

SCHEMBL7790301

CCC(C(N)=O)C1CCN(CCC2(c3ccc(C)c(C)c3)CCCN(C(=O)Cc3cc(Cl)cc(Cl)c3)C2)CC1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.45
TACR2 P21452 8/20 0.41
TACR1 P25103 7/20 0.41
HRH1 P35367 1/20 0.35
TACR3 P29371 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201066 0.85 CCR5 (0.45) CCR5TACR2TACR1HRH1TACR3
Hydrochloric Acid SCHEMBL6493645 0.85 CCR5 (0.45) CCR5TACR2TACR1HRH1TACR3
SCHEMBL5199609 0.83 TACR2 (0.43) CCR5TACR2TACR1TACR3
Hydrochloric Acid SCHEMBL6492132 0.82 TACR2 (0.42) CCR5TACR2TACR1TACR3
SCHEMBL6500864 0.80 EPHX2 (0.45) CCR5
SCHEMBL5200156 0.77 CCR5 (0.52) CCR5TACR2TACR1TACR3
SCHEMBL5201160 0.76 CCR5 (0.52) CCR5TACR2TACR1TACR3
Hydrochloric Acid SCHEMBL6490210 0.76 CCR5 (0.52) CCR5TACR2TACR1TACR3
SCHEMBL5203851 0.75 HSD11B1 (0.39) CCR5
SCHEMBL5200054 0.75 CCR5 (0.51) CCR5TACR2TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150970-A1 (1-PHENACY-3-PHENYL-3-PIPERIDYLETHYL)PIPERIDINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Sanofi-Aventis (FR) 2001-11-07 EP disclosed
WO-2000047572-A1 (1-PHENACY-3-PHENYL-3-PIPERIDYLETHYL)PIPERIDINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SANOFI-SYNTHELABO (FR) 2000-08-17 WO disclosed