SCHEMBL7791371

SCHEMBL7791371

CCCC(C=O)NC(=O)c1ccc(CSc2ccnc3cc(C(F)(F)F)ccc23)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.38
TAS1R1 Q7RTX1 2/20 0.38
CYP3A4 P08684 3/20 0.35
KMT2A Q03164 2/20 0.35
PRNP P04156 2/20 0.35
RXFP1 Q9HBX9 2/20 0.35
POLB P06746 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
KDR P35968 3/20 0.34
PRKD3 O94806 2/20 0.34
MAP4K4 O95819 2/20 0.34
GSK3A P49840 2/20 0.34
GSK3B P49841 2/20 0.34
AURKB Q96GD4 2/20 0.34
PRKD2 Q9BZL6 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
PLK4 O00444 1/20 0.34
DYRK3 O43781 1/20 0.34
CHEK2 O96017 1/20 0.34
FGFR1 P11362 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4881325 0.75 HDAC3 (0.44) KMT2APRNPRXFP1POLBSLC22A12
SCHEMBL4421777 0.73 MAPT (0.42) PRNPRXFP1SLC22A12KDRPRKD3
SCHEMBL28757760 0.72 RAC1 (0.38) KMT2APRNPRXFP1POLBMAPT
SCHEMBL7786986 0.69 KCNK2 (0.44) TAS1R3TAS1R1KMT2APRNPRXFP1
SCHEMBL4591807 0.67 RAC1 (0.52) KMT2APRNPRXFP1POLBSLC22A12
SCHEMBL20683281 0.66 RAC1 (0.54) KMT2APRNPRXFP1POLBSLC22A12
SCHEMBL27619323 0.66 DAO (0.39) KDRPRKD3MAP4K4GSK3AGSK3B
SCHEMBL4419754 0.66 DAO (0.39) KDRPRKD3MAP4K4GSK3AGSK3B
SCHEMBL25403102 0.64 RAC1 (0.52) KMT2APRNPRXFP1POLBSLC22A12
SCHEMBL27619372 0.64 RAC1 (0.41) CYP3A4KMT2APRNPRXFP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed