SCHEMBL7786986

SCHEMBL7786986

CCCC(C=O)NC(=O)c1ccc(CSc2ccc3ccccc3n2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK2 O95069 1/20 0.44
PRNP P04156 4/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
RAB9A P51151 3/20 0.42
RXFP1 Q9HBX9 4/20 0.42
MAPT P10636 4/20 0.42
KDM4E B2RXH2 3/20 0.42
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42
ALDH1A1 P00352 5/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPSR1 Q6W5P4 3/20 0.40
MAPK10 P53779 2/20 0.40
HDAC3 O15379 3/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC6 Q9UBN7 3/20 0.39
HDAC4 P56524 2/20 0.39
HDAC7 Q8WUI4 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789879 0.87 CAPN1 (0.48) KCNK2PRNPRAB9ARXFP1MAPT
SCHEMBL7789875 0.87 CAPN1 (0.48) KCNK2PRNPRAB9ARXFP1MAPT
SCHEMBL27676562 0.75 HDAC3 (0.53) KMT2AMEN1RAB9ATAS1R3TAS1R1
SCHEMBL11189080 0.75 RXFP1 (0.60) KCNK2PRNPKMT2AMEN1RAB9A
SCHEMBL27656629 0.74 RAB9A (0.54) KMT2AMEN1RAB9ATAS1R3TAS1R1
SCHEMBL1064818 0.72 HDAC1 (0.67) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL7787801 0.69 CAPN1 (0.58) KMT2AMEN1KDM4E
SCHEMBL7787804 0.69 CAPN1 (0.58) KMT2AMEN1KDM4E
SCHEMBL7791371 0.69 TAS1R3 (0.38) PRNPKMT2AMEN1RXFP1MAPT
SCHEMBL29177611 0.69 RXFP1 (0.60) PRNPKMT2AMEN1RAB9ARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed