SCHEMBL7793679

SCHEMBL7793679

CCCCOC(=O)COc1cccc(N)c1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.64
PPARA Q07869 3/20 0.54
PPARG P37231 2/20 0.54
PLA2G4B P0C869 3/20 0.52
CYP3A4 P08684 2/20 0.51
TP53 P04637 1/20 0.51
ALDH1A1 P00352 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
THRB P10828 1/20 0.47
FAAH O00519 1/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
PDE4D Q08499 1/20 0.46
SMPD1 P17405 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7801086 0.96 TSHR (0.71) TSHRPPARAPPARGPLA2G4BCYP3A4
SCHEMBL7802428 0.95 TSHR (0.74) TSHRPPARAPPARGPLA2G4BCYP3A4
SCHEMBL7801094 0.92 TSHR (0.59) TSHRPPARAPPARGPLA2G4BCYP3A4
SCHEMBL29577774 0.85 TP53 (0.62) TSHRPPARAPPARGCYP3A4TP53
SCHEMBL655678 0.85 TP53 (0.62) TSHRPPARAPPARGCYP3A4TP53
SCHEMBL109886 0.85 TSHR (0.86) TSHRCYP3A4TP53ALDH1A1CYP1A2
SCHEMBL27483976 0.84 CYP1A2 (0.59) TSHRPLA2G4BCYP3A4ALDH1A1TDP1
SCHEMBL202778 0.84 PLA2G4B (0.58) PPARAPPARGPLA2G4BALDH1A1TDP1
SCHEMBL31609710 0.84 PLA2G4B (0.58) PPARAPPARGPLA2G4BALDH1A1TDP1
SCHEMBL11655422 0.82 LTA4H (0.61) TSHRPLA2G4BFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900255-B1 DONOR-SUBSTITUTED OXINDIGO DERIVATIVES AND THEIR USE AS COLOURANTS CIBA SC HOLDING AG (CH) 2001-12-19 EP disclosed
US-6156914-A Donor-substituted oxindigo derivatives and their use as colorants CIBA SPECIALTY CHEMICALS CORPORATION (US) 2000-12-05 US disclosed
EP-0900255-A1 DONOR-SUBSTITUTED OXINDIGO DERIVATIVES AND THEIR USE AS COLOURANTS Ciba SC Holding AG (CH) 1999-03-10 EP disclosed
WO-1997041176-A1 DONOR-SUBSTITUTED OXINDIGO DERIVATIVES AND THEIR USE AS COLOURANTS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1997-11-06 WO disclosed