Bromide

Bromide

SCHEMBL7794743

Br.CCN1c2cc(O)ccc2C(C)=CC1(C)C

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
LMNA P02545 3/20 0.37
NPSR1 Q6W5P4 3/20 0.36
KMT2A Q03164 6/20 0.35
MEN1 O00255 5/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
POLB P06746 1/20 0.35
TSHR P16473 4/20 0.35
MAPK1 P28482 2/20 0.35
USP2 O75604 1/20 0.35
MCOLN3 Q8TDD5 1/20 0.34
KDM4E B2RXH2 6/20 0.34
MAPT P10636 4/20 0.34
GAA P10253 2/20 0.34
ALOX12 P18054 2/20 0.34
HSD17B10 Q99714 2/20 0.34
CASP1 P29466 1/20 0.33
HTT P42858 1/20 0.33
NPY1R P25929 1/20 0.32
RECQL P46063 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29430132 0.98 ALDH1A1 (0.42) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL20390457 0.87 ALDH1A1 (0.40) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL14850036 0.83 ALDH1A1 (0.54) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL3485083 0.81 ALDH1A1 (0.41) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL12388029 0.81 ALDH1A1 (0.40) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL29430125 0.78 ALDH1A1 (0.49) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL1917162 0.78 ALDH1A1 (0.49) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL15158277 0.77 ALDH1A1 (0.40) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL7801140 0.76 ALDH1A1 (0.40) ALDH1A1LMNANPSR1KMT2AMEN1
SCHEMBL15930651 0.76 TNF (0.42) ALDH1A1KMT2AMEN1L3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0962497-B1 Rhodamine derivates and their use in diagnostic systems ROCHE DIAGNOSTICS GMBH (DE) 2001-07-18 EP disclosed
US-6184379-B1 FLUORESCENT DYES USED IN DIAGNOSIS ROCHE DIAGNOSTICS GMBH (DE) 2001-02-06 US disclosed
EP-0962497-A1 Rhodamine derivates and their use in diagnostic systems Roche Diagnostics GmbH (DE) 1999-12-08 EP disclosed