SCHEMBL7795386

SCHEMBL7795386

COc1cc(C(NC(C)c2ccc(F)c(F)c2)c2ccc(F)cc2)cc(Nc2c(O)c(=O)c2=O)c1OC

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 5/20 0.39
IDO1 P14902 1/20 0.32
TDO2 P48775 1/20 0.32
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
PDE10A Q9Y233 3/20 0.31
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
MAPKAPK2 P49137 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7804313 0.94 CXCR2 (0.38) CXCR2IDO1TDO2CRHBPCRHR2
SCHEMBL7780384 0.87 CXCR2 (0.33) CXCR2MAPKAPK2
SCHEMBL7795456 0.85 CXCR2 (0.35) CXCR2GAAALDH1A1
SCHEMBL7787494 0.81 KMT2A (0.38) CXCR2CRHBPCRHR2GAAMAPT
Hydrochloric Acid SCHEMBL7801938 0.81 CXCR2 (0.35) CXCR2GAAMAPTSMN1; SMN2ALDH1A1
SCHEMBL7785125 0.81 CXCR2 (0.32) CXCR2
SCHEMBL7801984 0.81 CXCR2 (0.36) CXCR2IDO1MAPTMAPKAPK2MEN1
SCHEMBL7805393 0.79 CXCR2 (0.40) CXCR2MAPKAPK2MEN1KMT2A
SCHEMBL7795412 0.79 CXCR2 (0.40) CXCR2MAPKAPK2MEN1KMT2A
SCHEMBL7789230 0.79 KMT2A (0.36) CXCR2CRHBPCRHR2GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed