SCHEMBL7796074

SCHEMBL7796074

C=CCOc1ccc(-c2c(OC(C)C)cccc2C2=NC(C)(C)CO2)c(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SHMT2 P34897 1/20 0.35
ALDH1A1 P00352 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
PTPN1 P18031 2/20 0.33
KDM4E B2RXH2 1/20 0.32
MGAM O43451 3/20 0.32
GAA P10253 3/20 0.32
SI P14410 3/20 0.32
MGAM2 Q2M2H8 3/20 0.32
CD274 Q9NZQ7 1/20 0.31
NR3C1 P04150 1/20 0.31
PGR P06401 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
ALOX5 P09917 1/20 0.30
MAOB P27338 1/20 0.30
FGFR4 P22455 1/20 0.30
PDE10A Q9Y233 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7794735 0.89 KDM4E (0.37) ALDH1A1NPSR1PTPN1KDM4EHRH3
SCHEMBL8594056 0.88 SHMT2 (0.37) SHMT2ALDH1A1NPSR1KDM4EMGAM
SCHEMBL7794802 0.74 ALDH1A1 (0.43) ALDH1A1NPSR1PTPN1KDM4EMGAM
SCHEMBL6701333 0.71 PTPN1 (0.45) ALDH1A1PTPN1KDM4EGAA
SCHEMBL7786572 0.71 ALDH1A1 (0.41) ALDH1A1PTPN1KDM4EMGAMGAA
SCHEMBL7571712 0.71 PTPN1 (0.44) ALDH1A1PTPN1KDM4EGAA
SCHEMBL7792243 0.70 KDM4E (0.47) ALDH1A1NPSR1KDM4EHRH3
SCHEMBL7105642 0.68 KDM4E (0.47) ALDH1A1KDM4EHRH3
Iodide SCHEMBL7792207 0.68 CYP1A1 (0.36) ALDH1A1NPSR1KDM4EPDE10A
Iodide SCHEMBL7786337 0.68 CA1 (0.33) ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906268-B1 ALKYLOXYAMINO SUBSTITUTED FLUORENONES AND THEIR USE AS PROTEIN KINASE C INHIBITORS AVENTIS PHARMA INC (US) 2001-11-28 EP disclosed
US-6004959-A HYPOTENSIVE, ANTITUMOR, ANTIINFLAMMATORY AND ANTIASTHMATIC AGENTS; ANGIOGENESIS AND ALVEOLAR MACROPHAGE ACTIVATION INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed