SCHEMBL7798136

SCHEMBL7798136

c1ccc(CC2CCN(CCCn3ncc4cccc(-n5cnnc5)c43)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.50
SLC6A4 P31645 10/20 0.50
SLC6A3 Q01959 5/20 0.50
SIGMAR1 Q99720 2/20 0.47
CCR3 P51677 1/20 0.47
DRD4 P21917 2/20 0.47
KCNH2 Q12809 1/20 0.46
ADRB2 P07550 1/20 0.45
CHRM2 P08172 1/20 0.45
CHRM4 P08173 1/20 0.45
ADRB1 P08588 1/20 0.45
CHRM5 P08912 1/20 0.45
CHRM1 P11229 1/20 0.45
DRD2 P14416 1/20 0.45
CHRM3 P20309 1/20 0.45
ADRA1D P25100 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
DRD3 P35462 1/20 0.45
HTR1D P28221 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8031601 0.99 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3SIGMAR1CCR3
SCHEMBL7798184 0.85 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3SIGMAR1DRD4
Hydrochloric Acid SCHEMBL8021881 0.85 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3SIGMAR1DRD4
SCHEMBL7798221 0.79 HTR1D (0.55) SLC6A2SLC6A4SLC6A3SIGMAR1CCR3
Hydrochloric Acid SCHEMBL8031711 0.78 HTR1D (0.54) SLC6A2SLC6A4SLC6A3SIGMAR1CCR3
SCHEMBL7798285 0.76 SLC6A2 (0.50) SLC6A2SLC6A4SIGMAR1CCR3DRD4
Hydrochloric Acid SCHEMBL8021878 0.75 SLC6A2 (0.49) SLC6A2SLC6A4SIGMAR1CCR3DRD4
SCHEMBL5199674 0.70 CCR3 (0.74) SLC6A2SLC6A4SIGMAR1CCR3KCNH2
Hydrochloric Acid SCHEMBL8031614 0.69 HTR1A (0.41) SLC6A2SLC6A4SLC6A3SIGMAR1DRD4
SCHEMBL7807144 0.68 HTR1D (0.56) SLC6A2SLC6A4SIGMAR1CCR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902027-B1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR (FR) 2001-07-25 EP disclosed
EP-0902027-A1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-03-17 EP disclosed