SCHEMBL7798977

SCHEMBL7798977

CN1C(=O)CCC2c3cc(Cl)ccc3CCC21

nearest known ligand 0.80

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 20/20 0.80
SRD5A2 P31213 2/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7798978 1.00 SRD5A1 (0.80) SRD5A1SRD5A2
Bexlosteride SCHEMBL225679 0.89 SRD5A1 (1.00) SRD5A1SRD5A2
Bexlosteride SCHEMBL29569846 0.89 SRD5A1 (1.00) SRD5A1SRD5A2
Bexlosteride SCHEMBL7798944 0.89 SRD5A1 (1.00) SRD5A1SRD5A2
Bexlosteride SCHEMBL7194610 0.89 SRD5A1 (1.00) SRD5A1SRD5A2
Bexlosteride SCHEMBL13735634 0.89 SRD5A1 (1.00) SRD5A1SRD5A2
Bexlosteride SCHEMBL225678 0.89 SRD5A1 (1.00) SRD5A1SRD5A2
SCHEMBL7796407 0.83 SRD5A1 (0.66) SRD5A1SRD5A2
SCHEMBL7796412 0.83 SRD5A1 (0.66) SRD5A1SRD5A2
SCHEMBL7796276 0.83 SRD5A1 (0.71) SRD5A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0591583-B1 Benzo (f) quinolinones as 5-alpha-reductase inhibitors LILLY CO ELI (US) 2001-12-19 EP disclosed
EP-0532190-B1 Benzo(f)quinolinones as 5-alpha-reductase inhibitors LILLY CO ELI (US) 2000-12-27 EP disclosed
US-5541190-A TREATING BENIGN PROSTATIC HYPERPLASIA, MALE PATTERN BALDNESS, PROSTATIC CANCER, ANDROGENIC ALOPECIA ELI LILLY AND COMPANY (US) 1996-07-30 US disclosed
US-5495021-A STEROID 5 ALPHA-REDUCTASE INHIBITORS ELI LILLY AND COMPANY (US) 1996-02-27 US disclosed
US-5334767-A Steroid 5a-reductase inhibitor ELI LILLY AND COMPANY (US) 1994-08-02 US disclosed
EP-0591583-A1 Benzo (f) quinolinones as 5-alpha-reductase inhibitors ELI LILLY AND COMPANY (US) 1994-04-13 EP disclosed
US-5239075-A PROCESS FOR THE PREPARATION OF BENZO (F) QUINOLINONES ELI LILLY AND COMPANY (US) 1993-08-24 US disclosed
EP-0532190-A2 Benzo f quinolinones as 5-alpha-reductase inhibitors ELI LILLY AND COMPANY (US) 1993-03-17 EP disclosed