SCHEMBL7798995

SCHEMBL7798995

COc1ccc(CSC(C)(C)CC(N)(CN)CC(C)(C)SCc2ccc(OC)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
PRMT1 Q99873 1/20 0.46
IDO1 P14902 5/20 0.44
TAAR1 Q96RJ0 1/20 0.42
MAOB P27338 3/20 0.39
APP P05067 1/20 0.39
AGXT P21549 2/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
TSHR P16473 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16589112 0.86 IDO1 (0.47) CYP3A4CYP1A2CYP2D6PRMT1IDO1
SCHEMBL6578267 0.85 CYP3A4 (0.62) CYP3A4CYP1A2CYP2D6PRMT1IDO1
SCHEMBL20435360 0.80 TAAR1 (0.50) CYP3A4CYP1A2CYP2D6PRMT1IDO1
SCHEMBL11490965 0.77 IDO1 (0.51) CYP3A4CYP1A2CYP2D6PRMT1IDO1
SCHEMBL7668721 0.75 IDO1 (0.52) CYP3A4IDO1TAAR1MAOBAPP
SCHEMBL8376336 0.74 MEN1 (0.47) CYP3A4CYP1A2CYP2D6PRMT1IDO1
SCHEMBL27715705 0.74 IDO1 (0.45) CYP3A4IDO1TAAR1MAOBAPP
SCHEMBL7798992 0.74 TAAR1 (0.44) CYP3A4CYP1A2CYP2D6PRMT1IDO1
SCHEMBL30657036 0.74 TAAR1 (0.44) CYP3A4CYP1A2CYP2D6PRMT1IDO1
SCHEMBL4433692 0.73 TAAR1 (0.53) CYP3A4CYP1A2CYP2D6IDO1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750610-B1 PIPERIDYL-4-SUBSTITUTED THYROSINE DERIVATIVES AS SCINTIGRAPHIC IMAGING AGENTS FOR THE DIAGNOSIS OF THROMBOSIS DIATIDE INC (US) 2001-12-12 EP disclosed