SCHEMBL7800306

SCHEMBL7800306

CC(C)(C)OC(=O)NS(=O)(=O)NC[C@@H]1C[C@H](SC(c2ccccc2)(c2ccccc2)c2ccccc2)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.42
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
TDP1 Q9NUW8 1/20 0.37
MCL1 Q07820 3/20 0.36
ABCB1 P08183 1/20 0.36
ATM Q13315 1/20 0.36
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811544 0.87 CCR5 (0.41) CCR5TDP1ATM
SCHEMBL7805536 0.83 CA1 (0.43) CA12CA1ABCB1ATM
SCHEMBL10514723 0.82 CCR5 (0.43) CCR5TDP1ATM
SCHEMBL7806815 0.82 CCR5 (0.43) CCR5TDP1ATM
SCHEMBL7805543 0.82 TDP1 (0.43) CCR5TDP1ATM
SCHEMBL7805572 0.81 TDP1 (0.42) CCR5TDP1ATM
SCHEMBL9362971 0.81 TDP1 (0.40) CCR5TDP1ATM
SCHEMBL9366889 0.81 CCR5 (0.44) CCR5TDP1
SCHEMBL8782044 0.81 CCR5 (0.40) CCR5TDP1ATM
SCHEMBL8781845 0.81 CCR5 (0.40) CCR5TDP1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed