SCHEMBL7811544

SCHEMBL7811544

NS(=O)(=O)NC[C@@H]1C[C@H](SC(c2ccccc2)(c2ccccc2)c2ccccc2)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.41
TDP1 Q9NUW8 1/20 0.39
ATM Q13315 1/20 0.38
RAB9A P51151 3/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
NPC1 O15118 1/20 0.37
BCHE P06276 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8785254 0.90 CCR5 (0.40) CCR5TDP1ATMRAB9ACYP3A4
SCHEMBL7805572 0.87 TDP1 (0.42) CCR5TDP1ATMRAB9AMAPT
SCHEMBL7800306 0.87 CCR5 (0.42) CCR5TDP1ATM
SCHEMBL8781804 0.87 TDP1 (0.42) CCR5TDP1ATMRAB9AMAPT
SCHEMBL9138797 0.87 TDP1 (0.42) CCR5TDP1ATMRAB9AMAPT
SCHEMBL7805543 0.86 TDP1 (0.43) CCR5TDP1ATMRAB9AMAPT
SCHEMBL9362971 0.85 TDP1 (0.40) CCR5TDP1ATMRAB9AMAPT
SCHEMBL7806815 0.85 CCR5 (0.43) CCR5TDP1ATMRAB9A
SCHEMBL10514723 0.85 CCR5 (0.43) CCR5TDP1ATMRAB9A
SCHEMBL8782026 0.84 CCR5 (0.39) CCR5TDP1ATMRAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed