SCHEMBL7800514

SCHEMBL7800514

COc1ccc(CCN)cc1.O=Cc1ccc(Cl)cc1Cl

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.57
TDP1 Q9NUW8 1/20 0.54
MAOB P27338 7/20 0.53
IDO1 P14902 1/20 0.49
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7792891 0.89 TDP1 (0.57) TDP1MAOBIDO1MEN1KMT2A
SCHEMBL19497462 0.83 ALDH1A1 (0.49) TAAR1TDP1MEN1KMT2AALDH1A1
SCHEMBL7800146 0.79 TAAR1 (0.65) TAAR1TDP1MAOB
SCHEMBL4743206 0.78 ALDH1A1 (0.50) TDP1MEN1KMT2AALDH1A1RAB9A
SCHEMBL7801505 0.78 TAAR1 (0.57) TAAR1TDP1ALDH1A1
SCHEMBL7800221 0.77 TDP1 (0.53) TAAR1TDP1MAOBIDO1MEN1
SCHEMBL19497328 0.76 MEN1 (0.47) TAAR1TDP1MEN1KMT2AALDH1A1
SCHEMBL4634 0.75 TAAR1 (1.00) TAAR1MAOBIDO1
SCHEMBL14102978 0.74 NPC1 (0.61) TDP1MAOBMEN1KMT2AALDH1A1
Lysine SCHEMBL7798368 0.74 TDP1 (0.40) TDP1IDO1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed