SCHEMBL7801653

SCHEMBL7801653

COc1ccccc1N1CCN(CCCNc2c(C=O)c(=O)n(C)c(=O)n2C)CC1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 5/20 0.79
ADRA1D P25100 3/20 0.79
ADRA1B P35368 3/20 0.79
CYP3A4 P08684 2/20 0.79
ADRA2A P08913 2/20 0.79
ADRA2B P18089 2/20 0.79
ADRA2C P18825 2/20 0.79
PMP22 Q01453 2/20 0.79
HIF1A Q16665 1/20 0.79
HTR1A P08908 7/20 0.64
DRD2 P14416 5/20 0.64
DRD3 P35462 3/20 0.64
MAPT P10636 2/20 0.64
CYP2C9 P11712 2/20 0.64
CYP2C19 P33261 2/20 0.64
LMNA P02545 1/20 0.64
ADRB2 P07550 1/20 0.64
ADRB1 P08588 1/20 0.64
TSHR P16473 1/20 0.64
MAPK1 P28482 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7803659 0.89 ADRA1A (0.73) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
SCHEMBL7803666 0.89 ADRA1A (0.73) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
SCHEMBL7803792 0.89 ADRA1A (0.73) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
SCHEMBL7803794 0.89 ADRA1A (0.73) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
SCHEMBL6375436 0.88 ADRA1A (1.00) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
SCHEMBL7799623 0.87 ADRA1A (0.83) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
SCHEMBL7801661 0.81 ADRA1A (0.75) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
SCHEMBL14761169 0.80 ADRA1A (0.71) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
Urapidil SCHEMBL48992 0.78 HTR1A (1.00) ADRA1AADRA1DADRA1BCYP3A4ADRA2A
Urapidil SCHEMBL29363219 0.78 HTR1A (1.00) ADRA1AADRA1DADRA1BCYP3A4ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0796251-B1 URACIL DERIVATIVES BYK GULDEN LOMBERG CHEM FAB (DE) 2001-10-17 EP disclosed
US-6046329-A Uracil derivatives BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-04-04 US disclosed
EP-0796251-A1 URACIL DERIVATIVES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1997-09-24 EP disclosed
WO-1996017831-A1 URACIL DERIVATIVES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-06-13 WO disclosed