SCHEMBL7802249

SCHEMBL7802249

CS(=O)(=O)c1ccc(/C(=C2\CCOC2=O)c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.48
PTGS1 P23219 2/20 0.43
ABCB11 O95342 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MT-CO2 P00403 1/20 0.43
HTR1A P08908 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
MC4R P32245 1/20 0.43
ESR2 Q92731 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7887232 1.00 PTGS2 (0.48) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7802251 1.00 PTGS2 (0.48) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7807200 0.90 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL7807198 0.90 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL7807292 0.89 PTGS2 (0.48) PTGS2PTGS1ESR2
SCHEMBL1782770 0.89 PTGS2 (0.46) PTGS2PTGS1ADORA3
SCHEMBL6882900 0.89 AKR1C3 (0.42) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7806930 0.89 PTGS2 (0.46) PTGS2PTGS1ADORA3
SCHEMBL7807269 0.89 PTGS2 (0.48) PTGS2PTGS1ESR2
SCHEMBL6882905 0.89 AKR1C3 (0.42) PTGS2PTGS1ABCB11ALDH1A1MT-CO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971910-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS Merck Frosst Canada & Co. (CA) 2000-01-19 EP claimed
WO-1998043966-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA & CO. (CA) 1998-10-08 WO claimed
EP-0891345-B1 NOVEL FURAN DIARYLMETHYLIDENE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THERAPEUTICAL USES THEREOF UNION PHARMA SCIENT APPL (FR) 2001-08-16 EP disclosed
US-6180651-B1 ANTIINFLAMMATORY AGENTS; ANALGESICS BRISTOL-MYERS SQUIBB 2001-01-30 US disclosed
EP-0971910-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS Merck Frosst Canada & Co. (CA) 2000-01-19 EP disclosed
EP-0891345-A1 NOVEL FURAN DIARYLMETHYLIDENE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THERAPEUTICAL USES THEREOF LABORATOIRES UPSA (FR) 1999-01-20 EP disclosed
WO-1998043966-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA & CO. (CA) 1998-10-08 WO disclosed
WO-1997037984-A1 NOVEL FURAN DIARYLMETHYLIDENE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THERAPEUTICAL USES THEREOF LABORATOIRES UPSA (FR) 1997-10-16 WO disclosed