SCHEMBL7807200

SCHEMBL7807200

Cc1ccc(C(=C2CCOC2=O)c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.47
AKR1C3 P42330 1/20 0.41
PTGS1 P23219 3/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7807198 1.00 PTGS2 (0.47) PTGS2AKR1C3PTGS1NPC1RAB9A
SCHEMBL7802249 0.90 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL7802251 0.90 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL7887232 0.90 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL7808787 0.89 KMT2A (0.38) PTGS2PTGS1NPC1RAB9A
SCHEMBL7808789 0.89 KMT2A (0.38) PTGS2PTGS1NPC1RAB9A
SCHEMBL7807292 0.88 PTGS2 (0.48) PTGS2AKR1C3PTGS1
SCHEMBL7806930 0.88 PTGS2 (0.46) PTGS2AKR1C3PTGS1
SCHEMBL6882900 0.88 AKR1C3 (0.42) PTGS2AKR1C3PTGS1
SCHEMBL215270 0.88 CA1 (0.49) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891345-B1 NOVEL FURAN DIARYLMETHYLIDENE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THERAPEUTICAL USES THEREOF UNION PHARMA SCIENT APPL (FR) 2001-08-16 EP disclosed
US-6180651-B1 ANTIINFLAMMATORY AGENTS; ANALGESICS BRISTOL-MYERS SQUIBB 2001-01-30 US disclosed
WO-2000014082-A1 DIARYLMETHYLIDENE FURAN DERIVATIVES AS DRUGS WITH ANTI-INFLAMMATORY, ANALGESIC AND CHEMOPREVENTIVE PROPERTIES LABORATORIES UPSA (FR) 2000-03-16 WO disclosed