SCHEMBL7802833

SCHEMBL7802833

COc1cc(CN(C)C(=O)C(CCO)Cc2ccc(Cl)c(Cl)c2)cc(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.43
HSP90AA1 P07900 1/20 0.39
MAOB P27338 2/20 0.39
MAOA P21397 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CDK8 P49336 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
PNMT P11086 1/20 0.37
TSHR P16473 1/20 0.37
MCHR1 Q99705 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
TACR3 P29371 1/20 0.36
CCR2 P41597 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811353 0.91 MEN1 (0.46) MAOBSMN1; SMN2MEN1KMT2A
SCHEMBL7807793 0.86 TACR1 (0.42) TACR1HSP90AA1MAOBMAOAALDH1A1
SCHEMBL7815213 0.84 HPGD (0.48) TACR1HSP90AA1PNMTMEN1KMT2A
SCHEMBL7807547 0.83 KDM4E (0.44) HSP90AA1ALDH1A1HTTCDK8CLK4
SCHEMBL6973686 0.82 MEN1 (0.50) CDK8CLK4MEN1KMT2ATACR3
SCHEMBL7802970 0.82 TACR1 (0.50) TACR1
SCHEMBL7815381 0.81 KMT2A (0.41) HSP90AA1MAOBMAOACDK8CLK4
SCHEMBL7802956 0.79 TSHR (0.49) TACR1ALDH1A1HTTSMN1; SMN2TSHR
SCHEMBL7809519 0.77 MEN1 (0.45) MAOBSMN1; SMN2MEN1KMT2ATACR3
SCHEMBL7815536 0.76 SIGMAR1 (0.43) CDK8CLK4PNMTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-B1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2001-10-31 EP disclosed
US-5654316-A Piperidine derivatives as neurokinin antagonists SCHERING CORPORATION (US) 1997-08-05 US disclosed