SCHEMBL7811353

SCHEMBL7811353

COc1cccc(CN(C)C(=O)C(CCO)Cc2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
HSD17B2 P37059 4/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
DPP4 P27487 1/20 0.43
TAAR1 Q96RJ0 2/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
RECQL P46063 1/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
MAOB P27338 1/20 0.40
TSPO P30536 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7802833 0.91 TACR1 (0.43) MEN1KMT2ASMN1; SMN2MAOB
SCHEMBL7809519 0.87 MEN1 (0.45) MEN1KMT2AHSD17B2SMN1; SMN2DPP4
SCHEMBL7815213 0.86 HPGD (0.48) MEN1KMT2AHPGD
SCHEMBL7807547 0.83 KDM4E (0.44) MEN1KMT2AACHE
SCHEMBL6973686 0.82 MEN1 (0.50) MEN1KMT2ABCHEACHE
SCHEMBL7811517 0.80 ALDH1A1 (0.52) MEN1KMT2ASMN1; SMN2POLBHPGD
SCHEMBL7815381 0.79 KMT2A (0.41) MEN1KMT2APOLBMAOB
SCHEMBL7815536 0.78 SIGMAR1 (0.43) MEN1KMT2A
SCHEMBL7807793 0.77 TACR1 (0.42) MEN1KMT2ASMN1; SMN2MAOB
SCHEMBL7802970 0.77 TACR1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-B1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2001-10-31 EP disclosed
US-5654316-A Piperidine derivatives as neurokinin antagonists SCHERING CORPORATION (US) 1997-08-05 US disclosed