SCHEMBL7803589

SCHEMBL7803589

N#CC1(NC(=O)[C@H](CS(=O)(=O)Cc2ccc(F)cc2)N[C@@H](c2ccccc2)C(F)(F)F)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 1.00
CTSB P07858 14/20 1.00
CTSL P07711 14/20 1.00
CTSK P43235 10/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2816947 0.96 CTSS (0.93) CTSSCTSBCTSLCTSK
SCHEMBL3983009 0.95 CTSS (0.91) CTSSCTSBCTSLCTSK
SCHEMBL2821047 0.94 CTSL (0.89) CTSSCTSBCTSLCTSK
SCHEMBL2821048 0.94 CTSL (0.89) CTSSCTSBCTSLCTSK
SCHEMBL3417576 0.91 CTSS (0.83) CTSSCTSBCTSLCTSK
SCHEMBL2820622 0.90 CTSS (0.82) CTSSCTSBCTSLCTSK
SCHEMBL1271701 0.90 CTSS (0.81) CTSSCTSBCTSLCTSK
SCHEMBL1271702 0.90 CTSS (0.81) CTSSCTSBCTSLCTSK
SCHEMBL1272789 0.89 CTSS (0.81) CTSSCTSBCTSLCTSK
SCHEMBL2821335 0.89 CTSL (0.80) CTSSCTSBCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010148488-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS FOR THE TREATMENT OF VARIOUS DISEASES MERCK FROSST CANADA LTD. (CA) 2010-12-29 WO disclosed