SCHEMBL7804121

SCHEMBL7804121

c1ccc(CN2CCC(Cn3ccc4ccc(-n5cnnc5)cc43)C2)nc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 5/20 0.44
HTR1B P28222 5/20 0.44
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
BRD4 O60885 1/20 0.40
SIGMAR1 Q99720 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
DRD4 P21917 1/20 0.38
HRH1 P35367 1/20 0.37
LMNA P02545 1/20 0.37
KCNH2 Q12809 1/20 0.37
ALDH1A1 P00352 1/20 0.36
PDE2A O00408 1/20 0.36
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8031546 0.99 HTR1D (0.44) HTR1DHTR1BKDM4ESMN1; SMN2BRD4
SCHEMBL7804919 0.86 KDM4E (0.41) KDM4ESMN1; SMN2BRD4SIGMAR1L3MBTL1
SCHEMBL7804960 0.86 HTR1D (0.44) HTR1DHTR1BKDM4ESMN1; SMN2SIGMAR1
Hydrochloric Acid SCHEMBL8036973 0.85 KDM4E (0.41) KDM4ESMN1; SMN2BRD4SIGMAR1L3MBTL1
Hydrochloric Acid SCHEMBL8033560 0.85 HTR1D (0.43) HTR1DHTR1BKDM4ESMN1; SMN2SIGMAR1
SCHEMBL7804169 0.81 HTR1D (0.46) HTR1DHTR1BKDM4ESMN1; SMN2SIGMAR1
SCHEMBL7804076 0.81 HTR1D (0.44) HTR1DHTR1BKDM4ESIGMAR1ALDH1A1
Hydrochloric Acid SCHEMBL7805955 0.81 HTR1D (0.38) HTR1DHTR1B
Hydrochloric Acid SCHEMBL8021805 0.80 HTR1D (0.45) HTR1DHTR1BKDM4ESMN1; SMN2SIGMAR1
SCHEMBL7798125 0.80 HTR1D (0.56) HTR1DHTR1BKDM4EBRD4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902027-B1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR (FR) 2001-07-25 EP disclosed
EP-0902027-A1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-03-17 EP disclosed