SCHEMBL7804076

SCHEMBL7804076

c1coc(CN2CCC(Cn3ccc4ccc(-n5cnnc5)cc43)C2)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.44
HTR1B P28222 10/20 0.44
SIGMAR1 Q99720 1/20 0.36
ROCK2 O75116 1/20 0.35
CCR2 P41597 1/20 0.35
ROCK1 Q13464 1/20 0.35
GHSR Q92847 1/20 0.34
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
HTR1A P08908 1/20 0.33
HTR2A P28223 1/20 0.33
TRPV6 Q9H1D0 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8031070 0.99 HTR1D (0.44) HTR1DHTR1BSIGMAR1ROCK2CCR2
SCHEMBL7798179 0.81 HTR1D (0.46) HTR1DHTR1BHTR3EHTR3BHTR3A
SCHEMBL7804121 0.81 HTR1D (0.44) HTR1DHTR1BSIGMAR1ROCK2ROCK1
Hydrochloric Acid SCHEMBL7805955 0.81 HTR1D (0.38) HTR1DHTR1BHTR1AHTR2A
Hydrochloric Acid SCHEMBL8172775 0.80 HTR1D (0.45) HTR1DHTR1BSIGMAR1HTR3EHTR3B
Hydrochloric Acid SCHEMBL8031546 0.80 HTR1D (0.44) HTR1DHTR1BSIGMAR1ROCK2ROCK1
SCHEMBL7798296 0.80 HTR7 (0.40) HTR1DHTR1BHTR1AHTR2A
Hydrochloric Acid SCHEMBL8162484 0.79 HTR7 (0.40) HTR1DHTR1BHTR1AHTR2A
SCHEMBL7804089 0.79 HTR7 (0.44) SIGMAR1ALDH1A1
SCHEMBL7804162 0.77 HTR1D (0.45) HTR1DHTR1BSIGMAR1ROCK2CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902027-B1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR (FR) 2001-07-25 EP disclosed
EP-0902027-A1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-03-17 EP disclosed