SCHEMBL7804144

SCHEMBL7804144

c1ccc(N2CCN(CCCn3ccc4ccc(-n5cnnc5)cc43)CC2)nc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.50
POLB P06746 1/20 0.47
SLC6A4 P31645 2/20 0.46
SLC6A2 P23975 2/20 0.46
DRD3 P35462 6/20 0.45
DRD2 P14416 5/20 0.45
DRD4 P21917 4/20 0.45
HTR1A P08908 4/20 0.43
HTR2A P28223 4/20 0.43
HTR7 P34969 4/20 0.43
DRD1 P21728 4/20 0.43
ADRA2C P18825 3/20 0.43
HRH1 P35367 3/20 0.43
DRD5 P21918 2/20 0.43
SIGMAR1 Q99720 1/20 0.43
HTR1D P28221 2/20 0.43
HTR1B P28222 2/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA1D P25100 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8031163 0.99 KCNH2 (0.49) KCNH2POLBSLC6A4SLC6A2DRD3
SCHEMBL7806971 0.86 DRD3 (0.60) KCNH2DRD3DRD2DRD4HTR1A
SCHEMBL7798125 0.86 HTR1D (0.56) DRD3DRD2DRD4HRH1SIGMAR1
Hydrochloric Acid SCHEMBL8031131 0.85 DRD3 (0.59) KCNH2DRD3DRD2DRD4HTR1A
Hydrochloric Acid SCHEMBL8035289 0.85 HTR1D (0.55) DRD3DRD2DRD4HRH1SIGMAR1
SCHEMBL7805927 0.82 HTR7 (0.50) DRD3DRD2DRD4HTR7HTR1D
SCHEMBL7804093 0.81 HTR1D (0.54) DRD3DRD2DRD4HTR2ASIGMAR1
Hydrochloric Acid SCHEMBL8021825 0.81 HTR7 (0.49) DRD3DRD2DRD4HTR7HTR1D
Hydrochloric Acid SCHEMBL8021793 0.81 HTR1D (0.53) DRD3DRD2DRD4HTR2ASIGMAR1
SCHEMBL7805912 0.79 HTR1D (0.51) DRD3DRD2DRD4SIGMAR1HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902027-B1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR (FR) 2001-07-25 EP disclosed
EP-0902027-A1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-03-17 EP disclosed