SCHEMBL7804162

SCHEMBL7804162

c1coc(CN2CCC(n3ncc4ccc(-n5cnnc5)cc43)CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 3/20 0.45
HTR1B P28222 3/20 0.45
ROCK2 O75116 1/20 0.38
CCR2 P41597 1/20 0.38
ROCK1 Q13464 1/20 0.38
TRPV6 Q9H1D0 1/20 0.38
PARP1 P09874 2/20 0.36
CXCR3 P49682 2/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8036952 0.99 HTR1D (0.44) HTR1DHTR1BROCK2CCR2ROCK1
SCHEMBL7805945 0.83 DRD4 (0.49) HTR1DHTR1BALDH1A1KDM4EKMT2A
SCHEMBL7798179 0.83 HTR1D (0.46) HTR1DHTR1BTRPV6PARP1JAK2
Hydrochloric Acid SCHEMBL8037880 0.82 DRD4 (0.48) HTR1DHTR1BALDH1A1KDM4EKMT2A
Hydrochloric Acid SCHEMBL8172775 0.82 HTR1D (0.45) HTR1DHTR1BTRPV6PARP1JAK2
SCHEMBL7804112 0.79 CFTR (0.40) ROCK2CCR2ROCK1PARP1CXCR3
SCHEMBL7804158 0.77 HTR1B (0.50) HTR1DHTR1B
SCHEMBL7804076 0.77 HTR1D (0.44) HTR1DHTR1BROCK2CCR2ROCK1
Hydrochloric Acid SCHEMBL8021880 0.76 HTR1B (0.49) HTR1DHTR1B
Hydrochloric Acid SCHEMBL8031070 0.76 HTR1D (0.44) HTR1DHTR1BROCK2CCR2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902027-B1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR (FR) 2001-07-25 EP disclosed
EP-0902027-A1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-03-17 EP disclosed