SCHEMBL7804306

SCHEMBL7804306

C[C@@H](N)c1cc(F)c(F)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
TRPM8 Q7Z2W7 1/20 0.37
ADRB2 P07550 1/20 0.37
PDE2A O00408 2/20 0.36
DPP4 P27487 1/20 0.34
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
CA13 Q8N1Q1 1/20 0.31
AKT1 P31749 3/20 0.31
RPS6KA1 Q15418 3/20 0.31
PRKCA P17252 1/20 0.31
GRK2 P25098 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4087773 1.00 CES2 (0.39) CES2CES1TRPM8ADRB2PDE2A
SCHEMBL7795357 1.00 CES2 (0.39) CES2CES1TRPM8ADRB2PDE2A
Hydrochloric Acid SCHEMBL7787841 0.97 CES2 (0.38) CES2CES1TRPM8ADRB2PDE2A
Hydrochloric Acid SCHEMBL7787647 0.97 CES2 (0.38) CES2CES1TRPM8ADRB2PDE2A
SCHEMBL12563296 0.82 ADRB2 (0.36) TRPM8ADRB2PDE2ADPP4AKT1
SCHEMBL5380674 0.82 ADRB2 (0.39) ADRB2PDE2ADPP4
SCHEMBL19654073 0.82 ADRB2 (0.36) TRPM8ADRB2PDE2ADPP4AKT1
SCHEMBL5721005 0.82 ADRB2 (0.39) ADRB2PDE2ADPP4
SCHEMBL19654075 0.82 ADRB2 (0.36) TRPM8ADRB2PDE2ADPP4AKT1
SCHEMBL17041213 0.80 KDM1A (0.38) ADRB2PDE2ADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2681215-B1 SERINE/THREONINE KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2015-04-22 EP claimed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed