SCHEMBL7805563

SCHEMBL7805563

COC(=O)[C@H]1C[C@H](OS(C)(=O)=O)CN1C(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 4/20 0.48
ANPEP P15144 4/20 0.48
NR1H2 P55055 2/20 0.44
NR1H3 Q13133 1/20 0.44
PTPN1 P18031 1/20 0.42
P2RX3 P56373 1/20 0.39
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
UCHL1 P09936 1/20 0.36
MCL1 Q07820 5/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5058842 1.00 MMP2 (0.48) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL489252 1.00 MMP2 (0.48) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL699280 1.00 MMP2 (0.48) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL5691732 1.00 MMP2 (0.48) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL2252585 1.00 MMP2 (0.48) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL1154972 1.00 MMP2 (0.48) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL8607697 0.92 MMP2 (0.40) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL8609251 0.92 MMP2 (0.40) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL25436769 0.88 NR1H2 (0.43) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL19898506 0.88 NR1H2 (0.43) MMP2ANPEPNR1H2NR1H3PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023103523-A1 SUBSTITUTED BICYCLIC HETEROARYL COMPOUND AS KRAS G12D INHIBITOR 苏州浦合医药科技有限公司 2023-06-15 WO disclosed
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed