SCHEMBL7806830

SCHEMBL7806830

OCc1nc2cc(Oc3cccnc3)ccc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.49
LMNA P02545 2/20 0.49
CHEK2 O96017 1/20 0.43
CYP19A1 P11511 3/20 0.43
GRIN1 Q05586 2/20 0.41
GRIN2B Q13224 2/20 0.41
RHEB Q15382 1/20 0.39
LTA4H P09960 2/20 0.39
KDM4C Q9H3R0 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
ABL1 P00519 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
PPARG P37231 1/20 0.37
HTT P42858 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8524865 0.99 TDP1 (0.48) TDP1LMNACHEK2CYP19A1GRIN1
SCHEMBL7806832 0.90 CHEK2 (0.51) TDP1LMNACHEK2CYP19A1GRIN1
Hydrochloric Acid SCHEMBL8524871 0.89 CHEK2 (0.50) TDP1LMNACHEK2CYP19A1GRIN1
SCHEMBL7806900 0.85 GRIN1 (0.56) TDP1LMNAGRIN1GRIN2BRHEB
SCHEMBL7807032 0.84 TDP1 (0.43) TDP1LMNAGRIN1GRIN2BRHEB
Hydrochloric Acid SCHEMBL8480108 0.83 TDP1 (0.42) TDP1LMNAGRIN1GRIN2BRHEB
SCHEMBL28967661 0.80 LMNA (0.53) TDP1LMNACHEK2CYP19A1LTA4H
SCHEMBL30166989 0.80 LMNA (0.53) TDP1LMNACHEK2CYP19A1LTA4H
SCHEMBL7811234 0.80 GRIN1 (0.49) TDP1CHEK2GRIN1GRIN2BRHEB
Hydrochloric Acid SCHEMBL8478920 0.77 GRIN1 (0.47) TDP1LMNACHEK2GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820990-B1 Benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR (FR) 2001-01-17 EP disclosed
EP-0820990-A2 Novel benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR ET COMPAGNIE (FR) 1998-01-28 EP disclosed