SCHEMBL7807003

SCHEMBL7807003

CC(C)C(=O)OCC(O)(COC(=O)C(C)C)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
CYP2C9 P11712 2/20 0.46
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
CYP2C19 P33261 1/20 0.41
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
PTGS2 P35354 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MME P08473 1/20 0.39
ACE P12821 1/20 0.39
KIF11 P52732 2/20 0.38
DNMT1 P26358 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8152673 0.93 SMN1; SMN2 (0.43) MAPTALDH1A1POLBCYP2C9CYP1A2
SCHEMBL7809619 0.90 ALDH1A1 (0.51) MAPTALDH1A1POLBCYP2C9CYP1A2
SCHEMBL7813592 0.83 ALDH1A1 (0.48) MAPTALDH1A1POLBCYP2C9CYP1A2
SCHEMBL7808248 0.82 MAPT (0.61) MAPTALDH1A1POLBCYP2C9NPC1
SCHEMBL7810039 0.82 ALDH1A1 (0.50) MAPTALDH1A1POLBNPC1RAB9A
SCHEMBL7810773 0.81 GRIN2D (0.55) MAPTALDH1A1POLBCYP2C9CYP1A2
SCHEMBL7808224 0.81 ALDH1A1 (0.49) MAPTALDH1A1POLBGAANPC1
SCHEMBL7801779 0.79 ALDH1A1 (0.48) MAPTALDH1A1POLBKIF11
SCHEMBL7808447 0.79 ALDH1A1 (0.48) MAPTALDH1A1POLBGAARAB9A
SCHEMBL8148600 0.76 ALDH1A1 (0.49) MAPTALDH1A1POLBCYP2C9SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1120397-A2 Process for preparing triazole derivative KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2001-08-01 EP disclosed
EP-0704419-B1 PROCESS FOR PRODUCING AN OPTICALLY ACTIVE 2-ARYL-3-ACYLOXY-1,2-PROPANEDIOL KANEGAFUCHI CHEMICAL IND (JP) 2001-07-25 EP disclosed
US-6046354-A CHEMICAL INTERMEDIATES, E.G. 2-ARYL-1,3-DIACYLOXY-2-PROPANOL, FOR DRUGS AND FUNGICIDES,E.G. (R)-2-(2,4-DIFLUOROPHENYL)-3-(1H-1,2,4-TRIAZOLE-1-YL)-PROPANE-1,2-DIOL, KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2000-04-04 US disclosed
US-5840553-A OPTICALLY ACTIVE 2-ARYL-3-ACYLOXY-1,2,-PROPANE DIOL USING A MICROORGANISM OR ENZYME DERIVED FROM PORCINE PANCREAS; VIA STEREOSPECIFIC HYDROLYSIS OF A 2-ARYL-1,3-DIACYLOXY-2-PROPANOL; SYNTHETIC CHEMICAL INTERMEDIATES, FUNGICIDES KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1998-11-24 US disclosed
US-5654472-A OPTICALLY PURE 2-ARYL-3-ACYLOXY-1,2-PROPANEDIOL COMPOUNDS; CHEMICAL INTERMEDIATES KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1997-08-05 US disclosed
EP-0704419-A1 PROCESS FOR PRODUCING TRIAZOLE DERIVATIVE KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1996-04-03 EP disclosed