SCHEMBL7808447

SCHEMBL7808447

CC(C)C(=O)OCC(O)(COC(=O)C(C)C)c1ccc2ccccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
UGT2B7 P16662 1/20 0.40
PTPN1 P18031 1/20 0.40
KIF11 P52732 1/20 0.39
RECQL P46063 1/20 0.39
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PPARG P37231 2/20 0.38
PPARA Q07869 2/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
SLC6A2 P23975 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7809619 0.81 ALDH1A1 (0.51) ALDH1A1POLBMAPTKIF11RAB9A
SCHEMBL7807003 0.79 MAPT (0.47) ALDH1A1POLBMAPTKIF11GAA
SCHEMBL7801779 0.77 ALDH1A1 (0.48) ALDH1A1POLBMAPTKIF11RECQL
SCHEMBL7810039 0.76 ALDH1A1 (0.50) ALDH1A1POLBMAPTRECQLRAB9A
SCHEMBL7808248 0.76 MAPT (0.61) ALDH1A1POLBMAPTKIF11RAB9A
SCHEMBL7810773 0.75 GRIN2D (0.55) ALDH1A1POLBMAPTSMN1; SMN2MEN1
SCHEMBL7808224 0.75 ALDH1A1 (0.49) ALDH1A1POLBMAPTGAARAB9A
SCHEMBL7813592 0.74 ALDH1A1 (0.48) ALDH1A1POLBMAPTKIF11RAB9A
SCHEMBL7806844 0.73 ALDH1A1 (0.51) ALDH1A1POLBMAPTKIF11ADRB2
SCHEMBL8152673 0.73 SMN1; SMN2 (0.43) ALDH1A1POLBMAPTKIF11GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1120397-A2 Process for preparing triazole derivative KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2001-08-01 EP disclosed
EP-0704419-B1 PROCESS FOR PRODUCING AN OPTICALLY ACTIVE 2-ARYL-3-ACYLOXY-1,2-PROPANEDIOL KANEGAFUCHI CHEMICAL IND (JP) 2001-07-25 EP disclosed
US-6046354-A CHEMICAL INTERMEDIATES, E.G. 2-ARYL-1,3-DIACYLOXY-2-PROPANOL, FOR DRUGS AND FUNGICIDES,E.G. (R)-2-(2,4-DIFLUOROPHENYL)-3-(1H-1,2,4-TRIAZOLE-1-YL)-PROPANE-1,2-DIOL, KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2000-04-04 US disclosed
US-5840553-A OPTICALLY ACTIVE 2-ARYL-3-ACYLOXY-1,2,-PROPANE DIOL USING A MICROORGANISM OR ENZYME DERIVED FROM PORCINE PANCREAS; VIA STEREOSPECIFIC HYDROLYSIS OF A 2-ARYL-1,3-DIACYLOXY-2-PROPANOL; SYNTHETIC CHEMICAL INTERMEDIATES, FUNGICIDES KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1998-11-24 US disclosed
US-5654472-A OPTICALLY PURE 2-ARYL-3-ACYLOXY-1,2-PROPANEDIOL COMPOUNDS; CHEMICAL INTERMEDIATES KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1997-08-05 US disclosed
EP-0704419-A1 PROCESS FOR PRODUCING TRIAZOLE DERIVATIVE KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1996-04-03 EP disclosed