SCHEMBL7807384

SCHEMBL7807384

Cc1nccn1-c1ccc(COc2cccc(C3(C(N)=O)CCCC3)c2)cc1

nearest known ligand 0.66

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 11/20 0.66
GRM5 P41594 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7809136 0.98 ALOX5 (0.66) ALOX5GRM5
SCHEMBL7811098 0.96 ALOX5 (0.68) ALOX5GRM5
SCHEMBL7815083 0.92 ALOX5 (0.78) ALOX5
SCHEMBL8409170 0.88 ALOX5 (0.65) ALOX5GRM5
SCHEMBL8409097 0.87 ALOX5 (0.64) ALOX5GRM5
SCHEMBL7802752 0.87 ALOX5 (0.85) ALOX5GRM5
SCHEMBL8408893 0.86 ALOX5 (0.65) ALOX5GRM5
SCHEMBL7802468 0.86 ALOX5 (0.84) ALOX5GRM5
SCHEMBL8413029 0.84 ALOX5 (0.67) ALOX5GRM5
SCHEMBL2436940 0.79 ALOX5 (1.00) ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784054-B1 1,2,3,4-TETRAHYDROQUINOXALINEDIONE DERIVATIVES AND USE AS GLUTAMATE RECEPTOR ANTAGONISTS YAMANOUCHI PHARMA CO LTD (JP) 2001-11-28 EP disclosed
EP-0787127-B1 5-LIPOXYGENASE INHIBITORS PFIZER (US) 2001-01-03 EP disclosed
US-6096743-A 1,2,3,4-tetrahydroquinoxalinedione derivative YAMANOUCHI PHARMACEUTICALS CO., LTD. (JP) 2000-08-01 US disclosed
US-6063928-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS, CARDIOTONIC AGENTS PFIZER INC (US) 2000-05-16 US disclosed
EP-0784054-A1 1,2,3,4-TETRAHYDROQUINOXALINEDIONE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1997-07-16 EP disclosed