SCHEMBL7807777

SCHEMBL7807777

O=C(O)C(O)(CI)C(F)F

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CPT2 P23786 1/20 0.37
ACLY P53396 1/20 0.37
ODC1 P11926 1/20 0.33
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
BLM P54132 1/20 0.32
PMP22 Q01453 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6911619 0.75 CPT2 (0.37) CPT2ACLYODC1KDM4ELMNA
SCHEMBL6911617 0.75 CPT2 (0.37) CPT2ACLYODC1KDM4ELMNA
SCHEMBL6348790 0.64 ALDH1A1 (0.37) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL6913439 0.63 CPT2 (0.35) CPT2ACLY
SCHEMBL679467 0.62 ACLY (0.59) CPT2ACLYBLM
SCHEMBL29074266 0.62 ACLY (0.54) CPT2ACLYBLM
SCHEMBL17656832 0.62 ACLY (0.59) CPT2ACLYBLM
SCHEMBL4416232 0.62 ACLY (0.59) CPT2ACLYBLM
SCHEMBL31629798 0.62 ACLY (0.59) CPT2ACLYBLM
SCHEMBL18969113 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082110-A1 USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY AstraZeneca AB (SE) 2001-03-14 EP disclosed
WO-1999062506-A1 USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 1999-12-09 WO disclosed