SCHEMBL7807920

SCHEMBL7807920

Cn1cc(-c2cccnc2)c2cc(C=O)ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.50
GSK3B P49841 2/20 0.48
TTK P33981 1/20 0.47
SCN9A Q15858 1/20 0.46
CYP2A6 P11509 5/20 0.43
CYP2E1 P05181 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2B6 P20813 3/20 0.43
CYP2C19 P33261 3/20 0.43
NFATC1 O95644 1/20 0.43
DYRK1A Q13627 1/20 0.43
ERN1 O75460 3/20 0.41
ELANE P08246 1/20 0.40
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
CYP3A4 P08684 2/20 0.40
BRD4 O60885 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2A13 Q16696 1/20 0.38
CYP11B1 P15538 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7803219 0.76 CYP11B2 (0.64) NR4A2TTKCYP2A6CYP2E1CYP2C9
SCHEMBL21753339 0.74 TTK (0.51) TTKCYP2A6CYP2E1CYP2C9CYP2B6
SCHEMBL22159339 0.72 SCN9A (0.51) GSK3BSCN9ACYP2A6CYP3A4BRD4
SCHEMBL4241393 0.72 CYP11B2 (0.56) TTKCYP11B1CYP11B2
SCHEMBL3931286 0.71 TTK (0.49) TTKCYP2A6CYP2E1CYP2C9CYP2B6
SCHEMBL3933850 0.70 ERN1 (0.56) TTKERN1CYP3A4ALDH1A1CYP11B1
SCHEMBL23242341 0.70 CYP2A6 (0.50) CYP2A6ALDH1A1
SCHEMBL24296515 0.69 NR4A2 (0.76) NR4A2S1PR1S1PR3BRD4CYP11B1
SCHEMBL20914819 0.69 SCN9A (0.78) SCN9ACYP2C9CYP2B6CYP2C19
SCHEMBL18003572 0.68 PRMT5 (0.47) GSK3BDYRK1AELANEBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0949259-B1 N-HYDROXYUREA DERIVATIVES AND MEDICINAL COMPOSITIONS CONTAINING THE SAME NIKKEN CHEMICALS CO LTD (JP) 2001-06-20 EP disclosed
US-6184238-B1 ANTIALLERGENS, ANTIINFLAMMATORY AGENTS NIKKEN CHEMICALS CO., LTD. (JP) 2001-02-06 US disclosed
EP-0949259-A1 N-HYDROXYUREA DERIVATIVES AND MEDICINAL COMPOSITIONS CONTAINING THE SAME Nikken Chemicals Company, Limited (JP) 1999-10-13 EP disclosed