SCHEMBL7808323

SCHEMBL7808323

CN(C(=O)c1cc[c]cc1)c1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
KDM4E B2RXH2 2/20 0.44
KMT2A Q03164 2/20 0.44
RAB9A P51151 2/20 0.41
HSD17B10 Q99714 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
THRB P10828 1/20 0.41
TP53 P04637 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
LIPE Q05469 1/20 0.40
NPC1 O15118 1/20 0.40
HTT P42858 1/20 0.40
GRM1 Q13255 2/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
POLB P06746 1/20 0.40
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6316045 0.87 TSHR (0.58) TSHRKDM4EKMT2ARAB9AHSD17B10
SCHEMBL18765295 0.84 KDM4E (0.63) TSHRKDM4EKMT2ARAB9AHSD17B10
SCHEMBL7953771 0.84 TSHR (0.43) TSHRKDM4EKMT2ARAB9AHSD17B10
SCHEMBL3939111 0.81 TSHR (0.46) TSHRKDM4EKMT2ARAB9AHSD17B10
SCHEMBL7367970 0.81 TSHR (0.46) TSHRKDM4EKMT2ARAB9AHSD17B10
SCHEMBL5838645 0.77 HSD17B10 (0.60) TSHRKDM4ERAB9AHSD17B10TP53
SCHEMBL18765244 0.77 GAA (0.57) TSHRKMT2ARAB9AHSD17B10SMN1; SMN2
SCHEMBL7375901 0.77 MEN1 (0.64) KDM4EKMT2ARAB9ASMN1; SMN2TP53
SCHEMBL3895619 0.76 BRD4 (0.49) TSHRKDM4EKMT2ARAB9AHSD17B10
Hydrochloric Acid SCHEMBL18765408 0.76 GAA (0.56) TSHRKMT2ARAB9AHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed