SCHEMBL7808336

SCHEMBL7808336

COc1cncc(-c2ccc3c(nnn3CC(C)(C)C)c2Br)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 9/20 0.39
CYP11B2 P19099 9/20 0.39
CYP17A1 P05093 2/20 0.37
GRM2 Q14416 3/20 0.35
CYP3A4 P08684 2/20 0.35
SLC22A12 Q96S37 1/20 0.35
ALOX5AP P20292 2/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
PDE2A O00408 2/20 0.33
PDE10A Q9Y233 2/20 0.33
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
CYP1A1 P04798 1/20 0.31
CYP1B1 Q16678 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3475355 0.84 GRM2 (0.35) CYP11B1CYP11B2CYP17A1GRM2CYP3A4
SCHEMBL3476991 0.83 GRM2 (0.35) GRM2
SCHEMBL3475398 0.82 GRM2 (0.33) CYP11B1CYP11B2GRM2CYP1A2
SCHEMBL3475638 0.81 GRM2 (0.37) GRM2SLC22A12
SCHEMBL7816241 0.80 GRM2 (0.40) GRM2SLC22A12MKNK1MKNK2
SCHEMBL3469755 0.80 CNR1 (0.37) CYP11B1GRM2CYP3A4SLC22A12CYP1A2
SCHEMBL3475817 0.79 GRM2 (0.36) CYP17A1GRM2
SCHEMBL3474766 0.78 GRM2 (0.39) GRM2
SCHEMBL7819039 0.77 GRM2 (0.36) CYP17A1GRM2CYP3A4CYP1A2PDE2A
SCHEMBL7819300 0.76 GRM2 (0.39) GRM2CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed